Basic information Safety Supplier Related

Eprotirome

Basic information Safety Supplier Related

Eprotirome Basic information

Product Name:
Eprotirome
Synonyms:
  • eprotirome
  • N-[3,5-Dibromo-4-(4-hydroxy-3-isopropylphenoxy)phenyl]malonamic acid
  • 3-((3,5-Dibromo-4-(4-hydroxy-3-(1-methylethyl)phenoxy)phenyl)amino)-3-oxopropanoic acid
  • Kb-2115
  • Unii-958aq7B6R1
  • Propanoic acid,3-[[3,5-dibroMo-4-[4-hydroxy-3-(1-Methylethyl)phenoxy]phenyl]aMino]-3-oxo-
  • VPCSYAVXDAUHLT-UHFFFAOYSA-N
  • KB2115 Exclusive
CAS:
355129-15-6
MF:
C18H17Br2NO5
MW:
487.14
Mol File:
355129-15-6.mol
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Eprotirome Chemical Properties

Boiling point:
596.3±50.0 °C(Predicted)
Density 
1.708
storage temp. 
Sealed in dry,Room Temperature
solubility 
DMSO:84.0(Max Conc. mg/mL);172.43(Max Conc. mM)
DMF:30.0(Max Conc. mg/mL);61.58(Max Conc. mM)
Ethanol:63.5(Max Conc. mg/mL);130.35(Max Conc. mM)
Ethanol:PBS (pH 7.2) (1:1):0.5(Max Conc. mg/mL);1.03(Max Conc. mM)
form 
A crystalline solid
pka
3.16±0.32(Predicted)
color 
White to light yellow
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Eprotirome Usage And Synthesis

Uses

Eprotirome, is a liver-selective thyroid hormone receptor agonist.

in vivo

Eprotirome is a liver-selective thyroid hormone receptor agonist. Histological analysis of livers from mice treated with Eprotirome reveals that Eprotirome elicits a near complete elimination of lipid filled vacuoles that are characteristic of the livers from untreated control mice. Eprotirome treated mice also exhibit increased fasting glucose, but Eprotirome does not increase fasting insulin levels. Glucose levels of mice treated with Eprotirome continues to increase over time, leading to pronounced hyperglycemia by the end of the study. Temperature of mice treated with Eprotirome is decreased relative to untreated control mice[1].

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