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3,3a,7,7aα-Tetrahydro-3aα-hydroxy-2H-6-benzofuranone

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3,3a,7,7aα-Tetrahydro-3aα-hydroxy-2H-6-benzofuranone Basic information

Product Name:
3,3a,7,7aα-Tetrahydro-3aα-hydroxy-2H-6-benzofuranone
Synonyms:
  • 3,3a,7,7aα-Tetrahydro-3aα-hydroxy-2H-6-benzofuranone
  • (+)-Rengyolone
  • (3aS)-3,3a,7,7aβ-Tetrahydro-3aβ-hydroxybenzofura-6(2H)-one
  • (3aS)-3aβ-Hydroxy-2,3,3a,7aβ-tetrahydrobenzofuran-6(7H)-one
  • (3aS,7aS)-3,3a,7,7a-Tetrahydro-3a-hydroxy-2H-6-benzofuranone
  • Cleroindicin F
  • ent-Cleroindicin F
  • (3aR,7aR)-3,3a,7,7a-Tetrahydro-3a-hydroxy-6(2H)-benzofuranone
CAS:
189264-47-9
MF:
C8H10O3
MW:
154.16
Mol File:
189264-47-9.mol
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3,3a,7,7aα-Tetrahydro-3aα-hydroxy-2H-6-benzofuranone Chemical Properties

Boiling point:
332.9±42.0 °C(Predicted)
Density 
1.361±0.06 g/cm3(Predicted)
pka
12.88±0.20(Predicted)
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3,3a,7,7aα-Tetrahydro-3aα-hydroxy-2H-6-benzofuranone Usage And Synthesis

Uses

Cleroindicin F ((-)-Rengyolone), a cleroindicin, is an antimicrobial agent. Cleroindicin F shows relatively high anticandidal activity against Candida strains with a MIC value down to 12.5 μg/mL[1].

References

[1] Hasan Kirmizibekmez, et al. Secondary Metabolites from the Leaves of Digitalis viridiflora. Nat Prod Commun. 2017 Jan;12(1):59-61. PMID:30549826

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