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SULBENICILLIN

Product Name
SULBENICILLIN
CAS No.
41744-40-5
Chemical Name
SULBENICILLIN
Synonyms
SBPC;Kedacillina;Subenicillin;SULBENICILLIN;Sulbenicilina;(R)-Sulbenicillin;D-(-)-Sulbenicillin;Sulbenicillin, D-(-)-;a-Sulfobenzylpenicillin;SULBENICILLIN USP/EP/BP
CBNumber
CB6715306
Molecular Formula
C16H18N2O7S2
Formula Weight
414.45
MOL File
41744-40-5.mol
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SULBENICILLIN Property

Melting point:
197 °C (decomp)
Density 
1?+-.0.1 g/cm3(Predicted)
pka
0.28±0.50(Predicted)
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

American Custom Chemicals Corporation
Product number
API0013659
Product name
SULBENICILLIN
Purity
98.00%
Packaging
1G
Price
$1709.4
Updated
2021/12/16
AvaChem
Product number
2843
Product name
Sulbenicillin
Packaging
10mg
Price
$39
Updated
2021/12/16
AvaChem
Product number
2843
Product name
Sulbenicillin
Packaging
25mg
Price
$59
Updated
2021/12/16
AvaChem
Product number
2843
Product name
Sulbenicillin
Packaging
100mg
Price
$129
Updated
2021/12/16
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SULBENICILLIN Chemical Properties,Usage,Production

Originator

Lillacillin,Takeda,Japan,1973

Definition

ChEBI: A penicillin antibiotic having a 6beta-[phenyl(sulfo)acetamido] side-chain.

Manufacturing Process

To a suspension of 1.08 parts by weight of 6-aminopenicillanic acid in 8 parts by volume of water is added 1.48 parts by weight of sodium bicarbonate. After the mixture is dissolved, a solution of 1.18 parts by weight of α-sulfophenylacetyl chloride in 10 parts by volume of diethylether is gradually added thereto. The mixture is stirred at a temperature in the neighborhood of 0°C for 1 hour. The aqueous layer is washed twice with 10 parts by volume of portions of ether and adjusted to pH 1.2 with cation exchange resin of polystyrene sulfonic acid type under constant cooling. Then the solution is washed twice with 15 parts by volume of portions of ethyl acetate, followed by extraction twice with 15 parts by volume of portions of n-butanol. The extracts are combined and washed twice with 15 parts by volume of portions of water and, then, extracted with an aqueous solution of sodium bicarbonate. The extract is adjusted to pH 6.5, washed with ether and lyophilized to give the sodium salt of α-sulfobenzylpenicillin. Yield is 1.2 parts by weight.

Therapeutic Function

Antibacterial

Antimicrobial activity

α-Sulfobenzylpenicillin, a semisynthetic penicillin supplied as the disodium salt. Its antimicrobial spectrum and pharmacokinetic pharmacokinetic behavior closely resemble those of carbenicillin. Following intravenous administration of 4 g, the mean plasma concentration at 1 h was approximately 160 mg/L, with a plasma elimination half-life of around 70 min. It is largely excreted in the urine, about 80% of the dose appearing in the first 24 h, less than 5% as the penicilloic acid. It has been noted that the penicilloic acid causes much stronger platelet aggregation than its parent. It is of very limited availability.

SULBENICILLIN Preparation Products And Raw materials

Raw materials

Preparation Products

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SULBENICILLIN Suppliers

TargetMol Chemicals Inc.
Tel
+1-781-999-5354 +1-00000000000
Email
marketing@targetmol.com
Country
United States
ProdList
32165
Advantage
58
Amfinecom Inc.
Tel
--
Fax
--
Email
sales@amfinecom.com
Country
United States
ProdList
3062
Advantage
50
AmplaChem, Inc.
Tel
--
Fax
--
Email
info@amplacheminc.com
Country
United States
ProdList
428
Advantage
50
Ontario Chemicals, Inc
Tel
--
Fax
--
Email
info@ontariochem.com
Country
United States
ProdList
723
Advantage
50
Waterstone Technology, LLC
Tel
--
Fax
--
Email
sales@waterstonetech.com
Country
United States
ProdList
6786
Advantage
30
2A PharmaChem USA
Tel
--
Fax
--
Email
sales@2apharmachem.com
Country
United States
ProdList
6137
Advantage
39
3B Scientific Corporation
Tel
--
Fax
--
Email
sales@3bsc.com
Country
United States
ProdList
6718
Advantage
47
American Custom Chemicals Corporation
Tel
--
Fax
--
Email
sales@acccorporation.com
Country
United States
ProdList
6820
Advantage
51
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View Lastest Price from SULBENICILLIN manufacturers

Career Henan Chemical Co
Product
SULBENICILLIN 41744-40-5
Price
US $1.00/g
Min. Order
1g
Purity
≥98%
Supply Ability
g/kg/Ton
Release date
2019-12-25

41744-40-5, SULBENICILLINRelated Search:


  • SULBENICILLIN
  • Subenicillin
  • 4-Thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid, 3,3-dimethyl-7-oxo-6-[(phenylsulfoacetyl)amino]-, [2S-[2a,5a,6b(S*)]]-
  • 4-Thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid, 3,3-dimethyl-7-oxo-6-[[(2R)-phenylsulfoacetyl]amino]-, (2S,5R,6R)- (9CI)
  • a-Sulfobenzylpenicillin
  • D-(-)-Sulbenicillin
  • SBPC
  • Sulbenicillin, D-(-)-
  • (2S,5β)-3,3-Dimethyl-7-oxo-6α-[[(R)-phenyl(sulfo)acetyl]amino]-4-thia-1-azabicyclo[3.2.0]heptane-2β-carboxylic acid
  • (R)-Sulbenicillin
  • 6α-[(R)-Phenyl(sulfo)acetylamino]penicillanic acid
  • (2S,5R,6R)-6-((S)-Carbamoyl(phenyl)methanesulfonoyl)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid
  • (2S,5R,6R)-3,3-dimethyl-7-oxo-6-[(2-phenyl-2-sulfoacetyl)amino]-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid
  • (2S,5R,6R)-3,3-dimethyl-7-oxo-6-[(2-phenyl-2-sulfo-ethanoyl)amino]-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid
  • (2S,5R,6R)-7-keto-3,3-dimethyl-6-[(2-phenyl-2-sulfo-acetyl)amino]-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid
  • 4-Thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid, 3,3-dimethyl-7-oxo-6-[[(2R)-2-phenyl-2-sulfoacetyl]amino]-, (2S,5R,6R)-
  • SULBENICILLIN USP/EP/BP
  • Kedacillina
  • Sulbenicilina
  • 41744-40-5