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Nafcillin sodium salt monohydrate

Product Name
Nafcillin sodium salt monohydrate
CAS No.
7177-50-6
Chemical Name
Nafcillin sodium salt monohydrate
Synonyms
nafcillin sodium;Nafcillin sodium hydrate;Nafcillin sodium monohydrate;D00928;CL 8491;Unipen (tn);Naproxillin sodium;Emorfazone Impurity 1;Nafcillin sodium (usp);NAFCILLINSODIUMSTERILE
CBNumber
CB8769646
Molecular Formula
C21H25N2NaO6S
Formula Weight
456.49
MOL File
7177-50-6.mol
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Nafcillin sodium salt monohydrate Property

storage temp. 
2-8°C
solubility 
H2O: soluble50mg/mL
form 
A crystalline solid
color 
White to off-white
CAS DataBase Reference
7177-50-6(CAS DataBase Reference)
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Safety

Hazard Codes 
Xn
Risk Statements 
36/37/38-42/43
Safety Statements 
26-36-24/25
WGK Germany 
3
HS Code 
29411099
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Danger
Hazard statements

H315Causes skin irritation

H317May cause an allergic skin reaction

H319Causes serious eye irritation

H334May cause allergy or asthma symptoms or breathing difficulties if inhaled

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P284Wear respiratory protection.

P304+P340IF INHALED: Remove victim to fresh air and Keep at rest in a position comfortable for breathing.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P342+P311IF experiencing respiratory symptoms: call a POISON CENTER or doctor/physician.

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
N3269
Product name
Nafcillin sodium salt monohydrate
Packaging
5g
Price
$191
Updated
2024/03/01
Sigma-Aldrich
Product number
1450007
Product name
Nafcillin sodium
Purity
United States Pharmacopeia (USP) Reference Standard
Packaging
200mg
Price
$436
Updated
2024/03/01
Cayman Chemical
Product number
21008
Product name
Nafcillin (sodium salt hydrate)
Purity
≥95%
Packaging
1g
Price
$68
Updated
2024/03/01
Cayman Chemical
Product number
21008
Product name
Nafcillin (sodium salt hydrate)
Purity
≥95%
Packaging
5g
Price
$152
Updated
2024/03/01
Sigma-Aldrich
Product number
PHR1704
Product name
Nafcillin Sodium
Purity
Pharmaceutical Secondary Standard; Certified Reference Material
Packaging
1g
Price
$137
Updated
2022/05/15
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Nafcillin sodium salt monohydrate Chemical Properties,Usage,Production

Originator

Unipen,Wyeth,US,1964

Uses

Sodium Nafcillin Monohydrate is used as an antibiotic, used in the treatment, used in the treatment of gram-positive bacteria.

Uses

Antibacterial;Bacterial transpeptidase inhibitor

Uses

Nafcillin sodium salt monohydrate is an antibiotic resistant to beta-lactamase.

Definition

ChEBI: Nafcillin sodium monohydrate is an organic sodium salt and a hydrate. It contains a nafcillin sodium.

Manufacturing Process

A stirred suspension of 12.6 grams 6-aminopenicillanic acid in 130 ml dry alcohol-free chloroform was treated with 16 ml triethylamine and then with 13.8 grams of a solution of 2-ethoxy-1-naphthoyl chloride in 95 ml chloroform. After being washed successively with 58 ml each of 1 N and then 0.1 N hydrochloric acid the chloroform solution was extracted with N aqueous sodium bicarbonate (58 ml + 6 ml). The combined bicarbonate extracts were washed with 20 ml ether and then evaporated at low temperature and pressure to give the crude sodium salt of 2-ethoxy-1-naphthylpenicillin [also called sodium 6-(2-ethoxy-1-naphthamido)penicillinate] as a yellow powder (20.3 grams). This was dissolved in 20 ml water at 30°C and diluted with 180 ml n-butanol, also at 30°C, with stirring. Slow cooling to 0°C gave colorless needles of the product.

brand name

Nallpen (GlaxoSmithKline).

Therapeutic Function

Antibacterial

Clinical Use

Nafcillin sodium, 6-(2-ethoxy-1-naphthyl)penicillin sodium(Unipen), is another semisynthetic penicillin that resultedfrom the search for penicillinase-resistant compounds. Likemethicillin, nafcillin has substituents in positions ortho tothe point of attachment of the aromatic ring to the carboxamidegroup of penicillin. No doubt, the ethoxy group andthe second ring of the naphthalene group play steric roles instabilizing nafcillin against penicillinase. Very similar structureshave been reported to produce similar results in somesubstituted 2-biphenylpenicillins.
Unlike methicillin, nafcillin is stable enough in acid topermit its use by oral administration. When it is givenorally, its absorption is somewhat slow and incomplete,but satisfactory plasma levels may be achieved in about1 hour. Relatively small amounts are excreted throughthe kidneys; most is excreted in the bile. Even thoughsome cyclic reabsorption from the gut may occur, nafcillingiven orally should be readministered every 4 to 6 hours.This salt is readily soluble in water and may be administeredintramuscularly or intravenously to obtain highplasma concentrations quickly for the treatment of seriousinfections.
Nafcillin sodium may be used in infections causedsolely by penicillin G-resistant staphylococci or whenstreptococci are present also. Although it is recommendedthat it be used exclusively for such resistant infections, nafcillin is also effective against pneumococci and groupA -hemolytic streptococci. Because, like other penicillins,it may cause allergic side effects, it should be administeredwith care.

Nafcillin sodium salt monohydrate Preparation Products And Raw materials

Raw materials

Preparation Products

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Nafcillin sodium salt monohydrate Suppliers

CSPC Zhongnuo Pharmaceutical (Shijiazhuang) Co., Ltd.
Tel
0311-83092265
Fax
0311-83092288
Email
dongqj@mai.ecspc.com
Country
China
ProdList
24
Advantage
60
Shandong Xiya Chemical Co., Ltd
Tel
4009903999 13355009207
Fax
0539-6365991
Email
3007715519@qq.com
Country
China
ProdList
18738
Advantage
57
Sichuan Kulinan Technology Co., Ltd
Tel
400-1166-196 18981987031
Fax
028-84555506 800101999
Email
cdhxsj@163.com
Country
China
ProdList
11707
Advantage
57
Sinopharm Chemical Reagent Co,Ltd.
Tel
86-21-63210123
Fax
86-21-63290778 86-21-63218885
Email
sj_scrc@sinopharm.com
Country
China
ProdList
9815
Advantage
79
Beijing HuaMeiHuLiBiological Chemical
Tel
010-56205725
Fax
010-65763397
Email
waley188@sohu.com
Country
China
ProdList
12335
Advantage
58
Haoyuan Chemexpress Co., Ltd.
Tel
021-58950125
Fax
(86) 21-58955996
Email
info@chemexpress.com
Country
China
ProdList
7552
Advantage
61
Shanghai Aladdin Bio-Chem Technology Co.,LTD
Tel
400-400-6206333 18521732826
Fax
021-50323701
Email
market@aladdin-e.com
Country
China
ProdList
25003
Advantage
65
The future of Shanghai Industrial Co., Ltd.
Tel
021-61552785
Fax
021-55660885
Email
sales@shshiji.com
Country
China
ProdList
9545
Advantage
55
MedChemexpress LLC
Tel
021-58955995
Fax
609-228-5909
Email
sales@medchemexpress.cn
Country
United States
ProdList
4861
Advantage
58
Guangzhou Isun Pharmaceutical Co., Ltd
Tel
020-39119399 18927568969
Fax
020-39119999
Email
isunpharm@qq.com
Country
China
ProdList
4428
Advantage
55
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View Lastest Price from Nafcillin sodium salt monohydrate manufacturers

Hebei Mojin Biotechnology Co., Ltd
Product
Nafcillin sodium salt monohydrate 7177-50-6
Price
US $0.00/Kg/Bag
Min. Order
1KG
Purity
99%
Supply Ability
20ton
Release date
2021-04-25
Career Henan Chemical Co
Product
Nafcillin sodium salt monohydrate 7177-50-6
Price
US $3.00/KG
Min. Order
1KG
Purity
99%
Supply Ability
100kg
Release date
2019-08-07

7177-50-6, Nafcillin sodium salt monohydrateRelated Search:


  • Nafcillin monohydrate sodium salt
  • D00928
  • Nafcillin sodium (usp)
  • Nafcillin sodium monohydrate
  • Unipen (tn)
  • Nafcillin sodium salt monohydrate,6-(2-Ethoxy-1-naphthamido)penicillin
  • Nafcillin Sodium (200 mg)
  • Nafcillin sodiuM salt Monohydr
  • CL 8491
  • 4-Thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid, 6-[[(2-ethoxy-1-naphthalenyl)carbonyl]amino]-3,3-dimethyl-7-oxo-, sodium salt, hydrate (1:1:1), (2S,5R,6R)-
  • Nafcillin sodium hydrate
  • NAFCILLIN SODIUM SALT MONOHYDRATE
  • nafcillin sodium
  • 6-(2-ethoxy-1-naphthamido)penicillin
  • nafcillin sodium(Nafcillin sodium monohydrate)
  • Nafcillin sodium salt monohydrat
  • Sodium (2S,5R,6R)-6-[(2-ethoxynaphthalene-1-carbonyl)amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylate hydrate
  • NAFCILLINSODIUMSTERILE
  • Nafcillin (sodium salt hydrate)
  • Nafcillin sodium salt monohydrate USP/EP/BP
  • Nafcillin Sodium (1450007)
  • Naifcillin sodium monohydrate
  • Nafcillin sodium Powder USP Standard
  • Naproxillin sodium
  • Sodium (2S,5R,6R)-6-(2-ethoxy-1-naphthamido)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylate hydrate
  • Emorfazone Impurity 1
  • CL 8491|||nafcillin sodium
  • Nafcillin sodium hydrate in ACN:H2O (9:1)
  • 7177-50-6
  • C21H21N2O5SNaH2O
  • C21H23N2NaO6S
  • C21H21N2O5SH2ONa
  • C21H21N2NaO5SH2O
  • Antibiotics N-S
  • BioChemical
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