ChemicalBook > CAS DataBase List > 2-Iodo-4-nitroanisole

2-Iodo-4-nitroanisole

Product Name
2-Iodo-4-nitroanisole
CAS No.
5399-03-1
Chemical Name
2-Iodo-4-nitroanisole
Synonyms
2-Iodo-4-nitroanisol;2-Iodo-4-ntiroanisole;2-IODO-4-NITROANISOLE;2-iodo-4-nitrobenzyl ether;3-Iodo-4-methoxynitrobenzene;1-Iodo-2-Methoxy-5-nitrobenzene;2-IODO-1-METHOXY-4-NITROBENZENE;Benzene, 2-iodo-1-methoxy-4-nitro-;1,2-diaza-4-azanidacyclopenta-2,5-diene;3-Iodo-4-Methoxynitrobenzene[2-Iodo-4-nitroanisole]
CBNumber
CB9199754
Molecular Formula
C7H6INO3
Formula Weight
279.03
MOL File
5399-03-1.mol
More
Less

2-Iodo-4-nitroanisole Property

Melting point:
96-98°C
Boiling point:
343.3±27.0 °C(Predicted)
Density 
1.893±0.06 g/cm3(Predicted)
storage temp. 
Keep in dark place,Sealed in dry,Room Temperature
Appearance
Light brown to brown Solid
InChI
InChI=1S/C7H6INO3/c1-12-7-3-2-5(9(10)11)4-6(7)8/h2-4H,1H3
InChIKey
KBQBNJHOTNIGDD-UHFFFAOYSA-N
SMILES
C1(OC)=CC=C([N+]([O-])=O)C=C1I
CAS DataBase Reference
5399-03-1(CAS DataBase Reference)
More
Less

Safety

HS Code 
2909309090
More
Less

Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

More
Less

N-Bromosuccinimide Price

Sigma-Aldrich
Product number
S362816
Product name
2-IODO-4-NITROANISOLE
Purity
Aldrich<sup>CPR</sup>
Packaging
1 unit
Price
$185
Updated
2025/07/31
Sigma-Aldrich
Product number
S362816
Product name
2-IODO-4-NITROANISOLE
Purity
AldrichCPR
Packaging
250MG
Price
$179
Updated
2024/03/01
TRC
Product number
I737190
Product name
2-Iodo-4-nitroanisole
Packaging
1g
Price
$45
Updated
2021/12/16
TRC
Product number
I737190
Product name
2-Iodo-4-nitroanisole
Packaging
10g
Price
$75
Updated
2021/12/16
AK Scientific
Product number
X8330
Product name
2-Iodo-4-nitroanisole
Packaging
25g
Price
$77
Updated
2021/12/16
More
Less

2-Iodo-4-nitroanisole Chemical Properties,Usage,Production

Uses

2-Iodo-4-nitroanisole is commonly used in organic synthesis, especially as a synthetic intermediate in the fields of medicine and chemical research.

Synthesis

99-59-2

5399-03-1

Step A. Synthesis of 2-iodo-1-methoxy-4-nitrobenzene 2-Methoxy-5-nitroaniline (10.0 g, 0.060 mol) was suspended in water (150 mL) and concentrated sulfuric acid (12 mL, 0.22 mol) was added slowly. The temperature of the reaction mixture was maintained below 5 °C under cooling in an ice-salt bath, and a solution of sodium nitrite (4.8 g, 0.070 mol) in water (40 mL) was added dropwise. Subsequently, potassium iodide (16.8 g, 0.101 mol) was added and the mixture was heated to 90 °C and kept for 1 hour. Upon completion of the reaction, it was cooled to 0 °C and deep red crystals were precipitated, which were filtered, washed with water and dried. Purification by silica gel column chromatography (eluent: ethyl acetate/hexane) afforded the target compound 2-iodo-1-methoxy-4-nitrobenzene (13.6 g, 75% yield). 1H NMR (300 MHz, DMSO-d6): δ 8.57 (s, 1H), 8.28 (d, 1H), 7.19 (d, 1H), 3.98 (s, 3H). LCMS (M + H)+: m/z = 280.1 (C7H7INO3).

References

[1] Canadian Journal of Chemistry, 2005, vol. 83, # 3, p. 213 - 219
[2] Patent: US2009/286778, 2009, A1. Location in patent: Page/Page column 79
[3] Chem. News J. Ind. Sci., 1901, vol. 83, p. 285
[4] Journal of the Chemical Society, 1901, vol. 79, p. 1076,1077
[5] P. Ch. S., p. 238

2-Iodo-4-nitroanisole Preparation Products And Raw materials

Raw materials

Preparation Products

More
Less

2-Iodo-4-nitroanisole Suppliers

Nanjing Tangzheng Biomedical Technology Co., Ltd
Tel
13016839191
Email
719086845@qq.com
Country
China
ProdList
101
Advantage
58
J & K SCIENTIFIC LTD.
Tel
18210857532; 18210857532
Fax
86-10-82849933
Email
jkinfo@jkchemical.com
Country
China
ProdList
96815
Advantage
76
Energy Chemical
Tel
021-021-58432009 400-005-6266
Fax
021-58436166
Email
sales8178@energy-chemical.com
Country
China
ProdList
44801
Advantage
61
Wuhan Chemwish Technology Co., Ltd
Tel
86-027-67849912
Fax
86-027-87531808
Email
sales@chemwish.com
Country
China
ProdList
35896
Advantage
56
Capot Chemical Co., Ltd
Tel
+86 (0) 571 85 58 67 18
Fax
0086-571-85864795
Country
China
ProdList
18207
Advantage
66
Shanghai Sinch Parmaceuticals Tech. Co. Ltd.
Tel
+86-21-54098501
Fax
+86-21-54096319
Email
sales@sinch.com.cn
Country
China
ProdList
11598
Advantage
64
Shanghai Boc Chemical Co.,Ltd
Tel
021-34975603-808 18721111801
Fax
+86-21-34975602-805
Email
sales@bocpharma.com
Country
China
ProdList
1009
Advantage
64
Shanghai Longsheng chemical Co.,Ltd.
Tel
021-58099652-8005 13585536065
Fax
021-58099609
Email
bin.wu@shlschem.com
Country
China
ProdList
9883
Advantage
59
Shanghai Harvest Chemical Industrial Co., Ltd.
Tel
021-31038972,31038973 17321035817
Fax
+86-21-51385350
Email
sales@harvest-chem.com
Country
China
ProdList
2816
Advantage
64
China Langchem Inc.
Tel
0086-21-58956006
Fax
0086-21-58956100
Country
China
ProdList
7811
Advantage
57
More
Less

View Lastest Price from 2-Iodo-4-nitroanisole manufacturers

ZHENGZHOU JIUYI TIME NEW MATERIALS CO,.LTD
Product
2-Iodo-1-methoxy-4-nitrobenzene 5399-03-1
Price
US $2.00-5.00/KG
Min. Order
0.1KG
Purity
99%
Supply Ability
g-kg-tons
Release date
2025-07-10

5399-03-1, 2-Iodo-4-nitroanisoleRelated Search:


  • 2-IODO-4-NITROANISOLE
  • 2-Iodo-4-ntiroanisole
  • 1-Iodo-2-Methoxy-5-nitrobenzene
  • 2-Iodo-1-methoxy-4-nitrobenzene, 2-Iodo-4-nitrophenyl methyl ether
  • 3-Iodo-4-Methoxynitrobenzene[2-Iodo-4-nitroanisole]
  • 2-Iodo-4-nitroanisol
  • Benzene, 2-iodo-1-methoxy-4-nitro-
  • 2-IODO-1-METHOXY-4-NITROBENZENE
  • 1,2-diaza-4-azanidacyclopenta-2,5-diene
  • 3-Iodo-4-methoxynitrobenzene
  • 2-iodo-4-nitrobenzyl ether
  • 5399-03-1
  • 539-93-1
  • 1278045
  • 5399-3-1
  • 5933-03-1
  • C7H6INO3
  • C7H6NO3I
  • HALOGEN
  • Aromatic Ethers
  • Anisoles, Alkyloxy Compounds & Phenylacetates
  • Iodine Compounds
  • Nitro Compounds