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Boc-L-Cyclobutylglycine

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Boc-L-Cyclobutylglycine Basic information

Product Name:
Boc-L-Cyclobutylglycine
Synonyms:
  • 2-cyclobutyl-2-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]acetic acid
  • (2S)-2-{[(tert-butoxy)carbonyl]amino}-2-cyclobutylacetic acid
  • BOC-S-CYCBUGLY-OH
  • BOC-L-CYCLOBUTYL GLYCINE
  • BOC-(2S)-GLY(2-CYCLOBUTYL)
  • (S)-TERT-BUTOXYCARBONYLAMINO-CYCLOBUTYL-ACETIC ACID
  • (S)-N-ALPHA-T-BUTYLOXYCARBONYL-CYCLOBUTYLGLYCINE
  • BOC-L-CYCLOBUTYLGLYCINE 98%
CAS:
155905-77-4
MF:
C11H19NO4
MW:
229.27
EINECS:
200-110-4
Product Categories:
  • pharmacetical
Mol File:
155905-77-4.mol
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Boc-L-Cyclobutylglycine Chemical Properties

Boiling point:
379.1±25.0 °C(Predicted)
Density 
1.169±0.06 g/cm3(Predicted)
storage temp. 
Sealed in dry,Room Temperature
pka
4.06±0.10(Predicted)
form 
Solid
color 
White to off-white
optical activity
3°(C=0.01g/ml MEOH)
InChI
InChI=1/C11H19NO4/c1-11(2,3)16-10(15)12-8(9(13)14)7-5-4-6-7/h7-8H,4-6H2,1-3H3,(H,12,15)(H,13,14)/t8-/s3
InChIKey
OHDFGIXTRBDGRB-SBYBRXNCNA-N
SMILES
C(=O)(OC(C)(C)C)N[C@@H](C1CCC1)C(O)=O |&1:8,r|
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Safety Information

HS Code 
2924297099
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Boc-L-Cyclobutylglycine Usage And Synthesis

Uses

Boc-L-cyclobutylglycine is a glycine derivative that can be used for PI3K inhibitor synthesis[1].

References

[1] Kim YS, et al. Synthesis and biological evaluation of novel purinyl quinazolinone derivatives as PI3Kδ-specific inhibitors for the treatment of hematologic malignancies. Bioorg Med Chem. 2021 Sep 1;45:116312. DOI:10.1016/j.bmc.2021.116312

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