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6-(Trifluoromethyl)nicotinic acid

Product Name
6-(Trifluoromethyl)nicotinic acid
CAS No.
231291-22-8
Chemical Name
6-(Trifluoromethyl)nicotinic acid
Synonyms
3,5-Dichloropyrazine-2-carboxylic acid;6-(Trifluoromethyl)-3-pyridinecarboxylic acid;6-(TrifL;6-Trifluoromethyl;RARECHEM AL BO 1001;6-(TRIFLUOROMETHYL)PYRIDI;6-Trifluoromethylnicotic acid;TRIFLUOROMETHYL NICOTINIC ACID;6-(TRIFLUROMETHYL)NICOTINICACID;6- threefluorine Methylnicotinate
CBNumber
CB3440751
Molecular Formula
C7H4F3NO2
Formula Weight
191.11
MOL File
231291-22-8.mol
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6-(Trifluoromethyl)nicotinic acid Property

Melting point:
193-197 °C(lit.)
Boiling point:
259.3±40.0 °C(Predicted)
Density 
1.484±0.06 g/cm3(Predicted)
storage temp. 
Inert atmosphere,Room Temperature
solubility 
Acetonitrile (Slightly), Methanol (Slightly)
form 
Solid
pka
2.96±0.10(Predicted)
color 
Pale Beige to Light Brown
InChI
InChI=1S/C7H4F3NO2/c8-7(9,10)5-2-1-4(3-11-5)6(12)13/h1-3H,(H,12,13)
InChIKey
JNYLMODTPLSLIF-UHFFFAOYSA-N
SMILES
C1=NC(C(F)(F)F)=CC=C1C(O)=O
CAS DataBase Reference
231291-22-8(CAS DataBase Reference)
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Safety

Hazard Codes 
Xi
Risk Statements 
36/37/38
Safety Statements 
26-36
WGK Germany 
3
HazardClass 
IRRITANT
HS Code 
29333990
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P304+P340IF INHALED: Remove victim to fresh air and Keep at rest in a position comfortable for breathing.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P405Store locked up.

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N-Bromosuccinimide Price

TCI Chemical
Product number
T2203
Product name
6-(Trifluoromethyl)nicotinic Acid
Purity
>98.0%(GC)
Packaging
1g
Price
$34
Updated
2025/07/31
TCI Chemical
Product number
T2203
Product name
6-(Trifluoromethyl)nicotinic Acid
Purity
>98.0%(GC)
Packaging
5g
Price
$135
Updated
2025/07/31
TRC
Product number
T790650
Product name
6-(Trifluoromethyl)nicotinic Acid
Packaging
10g
Price
$45
Updated
2021/12/16
TRC
Product number
T790650
Product name
6-(Trifluoromethyl)nicotinic Acid
Packaging
25g
Price
$85
Updated
2021/12/16
Frontier Specialty Chemicals
Product number
T11123
Product name
6-(Trifluoromethyl)nicotinic Acid
Purity
98%
Packaging
1g
Price
$4
Updated
2021/12/16
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6-(Trifluoromethyl)nicotinic acid Chemical Properties,Usage,Production

Physical properties

6-Trifluoromethylnicotinic acid is a white powder with a melting point of 193-197 °C. It has a boiling point of 259.3℃ at 760 mmHg. Its density is 1.484 g/cm3. Its flash point, refractive index and vapor pressure are 110.6℃, 1.475 and 0.007mmHg at 25°C, respectively.

Uses

6-Trifluoromethyl Nicotinic Acid can be prepared to use Raf inhibitors to treat cancer.

Synthesis

216431-85-5

231291-22-8

To a 10L three-necked flask were added 1420 g of water, 2440 g of sulfuric acid, and 150 mL of glacial acetic acid, and 870 g (5 mol) of 6-(trifluoromethyl)nicotinonitrile was added slowly. The mixture was heated to reflux and kept overnight. Upon completion of the reaction, the reaction mixture was cooled, ice was added and the mixture was cooled using ice brine to precipitate a white solid. After filtration, the filtrate was extracted with ethyl acetate. The organic phases were combined and washed twice with water, followed by drying the organic phase to acidity. After washing, 930 g of 6-(trifluoromethyl)-3-pyridinecarboxylic acid was obtained as a beige solid in 97.3% yield.

References

[1] Patent: CN107298677, 2017, A. Location in patent: Paragraph 0036-0038
[2] Patent: CN107337638, 2017, A. Location in patent: Paragraph 0031; 0032; 0033
[3] Patent: EP1122242, 2001, A1
[4] Patent: US6673799, 2004, B1. Location in patent: Page column 16

6-(Trifluoromethyl)nicotinic acid Preparation Products And Raw materials

Raw materials

Preparation Products

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6-(Trifluoromethyl)nicotinic acid Suppliers

Shanghai Weiyuan Technology Co., Ltd.
Tel
13024122785 17356341931
Email
sales@shweiyuan.cn
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China
ProdList
280
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Nanjing YiFan Biological Technology Co., Ltd.
Tel
025-025-52700520 18914499889
Fax
025-52700520
Email
sales@yfbiotech.com
Country
China
ProdList
495
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58
Changzhou Huanling Chemical Co., Ltd.
Tel
0519-89803565 13776850645
Fax
0519-89803575
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info4@huanlingchem.com
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China
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Shanghai Fei Yan Chemical Technology Co., Ltd.
Tel
021-34663897 13816465839
Fax
021-34663897
Email
1141976404@qq.com
Country
China
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Beijing Sintong Pharma Technology Co., Ltd.
Tel
13466647005 13466647005;
Email
47652055@qq.com
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China
ProdList
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Hangzhou Copiore Chemical Co., Ltd.
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0571-56501939;0571-56076030 13757145729
Fax
0571-56501939
Email
sales@copiore.com
Country
China
ProdList
299
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J & K SCIENTIFIC LTD.
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18210857532; 18210857532
Fax
86-10-82849933
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jkinfo@jkchemical.com
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China
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96815
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PharmaBlock Sciences (Nanjing),Inc.
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025-86918202 4000255188
Fax
86-025-86918232
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sales@pharmablock.com
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China
ProdList
5000
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55
Meryer (Shanghai) Chemical Technology Co., Ltd.
Tel
4006356688 18621169109
Fax
86-21-61259102
Email
market03@meryer.com
Country
China
ProdList
40228
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62
INTATRADE GmbH
Tel
+49 3493/605464
Fax
+49 3493/605470
Email
sales@intatrade.de
Country
Germany
ProdList
3572
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View Lastest Price from 6-(Trifluoromethyl)nicotinic acid manufacturers

Hebei Chuanghai Biotechnology Co., Ltd
Product
6-(Trifluoromethyl)nicotinic acid 231291-22-8
Price
US $1.00/KG
Min. Order
1KG
Purity
99%
Supply Ability
10 mt
Release date
2024-10-24
Hebei Zhuanglai Chemical Trading Co Ltd
Product
6-(Trifluoromethyl)nicotinic acid 231291-22-8
Price
US $10.00/kg
Min. Order
1kg
Purity
99%
Supply Ability
20 ton
Release date
2024-12-18
Henan Aochuang Chemical Co.,Ltd.
Product
6-(Trifluoromethyl)nicotinic acid 231291-22-8
Price
US $0.00-0.00/KG
Min. Order
1KG
Purity
98%
Supply Ability
1Ton
Release date
2022-10-12

231291-22-8, 6-(Trifluoromethyl)nicotinic acidRelated Search:


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