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FILGRASTIM

Product Name
FILGRASTIM
CAS No.
121181-53-1
Chemical Name
FILGRASTIM
Synonyms
Figrastim;FILGRASTIM;Filgrastim CRS;FILGRASTIM USP/EP/BP;Filgrastim DISCONTINUED;filgrastimconcentratedSolution;n-l-methionyl-colony-stimulatingfactor(humanclone1034;Filgrastim for Bioassay (96,815 IU) (COLD SHIPMENT REQUIRED);Filgrastim System Suitability (COLD SHIPMENT REQUIRED) (1 mg);Colony-stiMulating factor (huMan clone 1034), N-L-Methionyl- (9CI)
CBNumber
CB6324250
Molecular Formula
W99
Formula Weight
0
MOL File
Mol file
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FILGRASTIM Property

storage temp. 
-70°C
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Safety

HS Code 
3002905150
Hazardous Substances Data
121181-53-1(Hazardous Substances Data)
Toxicity
LD50 oral in rat: > 3mg/kg
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H361Suspected of damaging fertility or the unborn child

Precautionary statements

P201Obtain special instructions before use.

P202Do not handle until all safety precautions have been read and understood.

P281Use personal protective equipment as required.

P308+P313IF exposed or concerned: Get medical advice/attention.

P405Store locked up.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
Y0001173
Product name
Filgrastim
Purity
European Pharmacopoeia (EP) Reference Standard
Packaging
y0001173
Price
$220
Updated
2024/03/01
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FILGRASTIM Chemical Properties,Usage,Production

Description

Filgrastim is a recombinant human granulocyte colony stimulating factor (G-CSF) indicated as an adjunct to cancer chemotherapy for patients with non-myeloid malignancies. It reduces the duration of chemotherapy-induced neutropenia by forcing immature leucocytes to differentiate into neutrophils, thereby decreasing the incidence and length of infections.Bone pain is the most significant side effect.Chugai launched the second G-CSF, lenograstim, in December 1991. Other potential uses include bone marrow transplants, myelodysplastic syndromes and febrilelchronic neutropenia.

Chemical Properties

Clear, colourless or slightly yellowish liquid

Originator

Amgen (U.S.A.)

Uses

Antineutropenic; hematopoietic stimulant.

Uses

Filgrastim is a human granulocyte colony stimulating factor (G-CSF) used to treat neutropenia.

Indications

Filgrastim (Neupogen) is a human recombinant granulocyte colony–stimulating factor (rG-CSF) produced using recombinant DNA technology. It acts on precursor hematopoietic cells in the bone marrow by binding to specific receptors that stimulate cellular proliferation and differentiation into neutrophils. It also enhances some neutrophil functions, including phagocytosis and antibody-dependent killing.

brand name

Neupogen (Amgen).

Clinical Use

Filgrastim, G-CSF, Neupogen, stimulates the proliferation ofgranulocytes (especially neutrophils) by mobilizinghematopoietic stem cells in the bone marrow. The native protein is glycosylated.Filgrastim selectively stimulates proliferation and differentiationof neutrophil precursors in the bone marrow. Thisleads to the release of mature neutrophils into the circulationfrom the bone marrow. Filgrastim also affects mature neutrophilsby enhancing phagocytic activity, priming the cellularmetabolic pathways associated with the respiratoryburst, enhancing antibody-dependent killing, and increasingthe expression of some functions associated with cell surfaceantigens.
In patients receiving chemotherapy with drugs such ascyclophosphamide, doxorubicin, and etoposide, the incidenceof neutropenia accompanied by fever is rather high.Administration of G-CSF reduces the time of neutrophilrecovery and duration of fever in adults with acute myelogenousleukemia. The number of infections, days thatantibiotics are required, and duration of hospitalization arealso reduced.

Clinical Use

Filgrastim is used to accelerate recovery of neutrophils after chemotherapy, both to prevent infections and to shorten the duration of neutropenia in patients in whom infections have developed.

Side effects

The drug is generally well tolerated, with the major adverse reaction being mild to moderate bone pain secondary to stimulation of bone marrow proliferation.

Veterinary Drugs and Treatments

Filgrastim may be of benefit in treating neutropenias in dogs or cats when the intrinsic response to endogenously produced cytokines is thought to be inadequate and there is evidence that there are precursors in the bone marrow available. Because of the drug’s cost and lack of good evidence for its efficacy in reducing mortality versus using antibiotic therapy alone, its use in small animal medicine is somewhat controversial.

Drug interactions

Potentially hazardous interactions with other drugs
Cytotoxics: neutropenia possibly exacerbated with capecitabine, fluorouracil and tegafur.

Metabolism

Filgrastim is primarily eliminated by the kidney and neutrophils/neutrophil precursors; the latter presumably involves binding of the growth factor to the G-CSF receptor on the cell surface, internalisation of the growth factor-receptor complexes via endocytosis, and subsequent degradation inside the cells

FILGRASTIM Preparation Products And Raw materials

Raw materials

Preparation Products

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FILGRASTIM Suppliers

Hangzhou Sage Chemical Co., Ltd.
Tel
+86057186818502 13588463833
Fax
Pls mail us for more information!
Email
info@sagechem.com
Country
China
ProdList
10266
Advantage
58
Beijing HuaMeiHuLiBiological Chemical
Tel
010-56205725
Fax
010-65763397
Email
waley188@sohu.com
Country
China
ProdList
12335
Advantage
58
Chizhou Kailong Import and Export Trade Co., Ltd.
Tel
Fax
-
Email
xg01_gj@163.com
Country
China
ProdList
9484
Advantage
50
Shanghai Synchem Pharma Co., ltd
Tel
21-619849051-1 18521059765
Email
synchempharma@aliyun.com
Country
China
ProdList
6463
Advantage
55
Beijing Solarbio Science & Tecnology Co., Ltd.
Tel
010-50973186 4009686088
Email
3193328036@qq.com
Country
China
ProdList
18338
Advantage
68
Alchemist-pharm chemical Technology Co. Ltd.
Tel
0371-67991738 13783628208
Fax
QQ 412703949
Email
carl@alchemist-pharm.com
Country
China
ProdList
1872
Advantage
58
Hebei Zhanyao Biotechnology Co. Ltd
Tel
15369953316 +8615369953316
Email
admin@zhanyaobio.com
Country
China
ProdList
2123
Advantage
58
Dideu Industries Group Limited
Tel
+86-29-89586680 +86-15129568250
Email
1026@dideu.com
Country
China
ProdList
22883
Advantage
58
AFINE CHEMICALS LIMITED
Tel
+86-0571-85134551
Fax
008657185134895
Email
sales@afinechem.com
Country
China
ProdList
15354
Advantage
58
Chemwill Asia Co.,Ltd.
Tel
86-21-51086038
Fax
86-21-51861608
Email
chemwill_asia@126.com
Country
CHINA
ProdList
23912
Advantage
58
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View Lastest Price from FILGRASTIM manufacturers

BEIJING SJAR TECHNOLOGY DEVELOPMENT CO., LTD.
Product
Filgrastim 121181-53-1
Price
US $0.00/g
Min. Order
1g
Purity
More Than 99%
Supply Ability
100kg/Month
Release date
2024-10-16
Hebei Zhanyao Biotechnology Co. Ltd
Product
FILGRASTIM 121181-53-1
Price
US $10.00/Kg/Bag
Min. Order
1Kg/Bag
Purity
99%
Supply Ability
20 Tons
Release date
2021-11-22
Dideu Industries Group Limited
Product
FILGRASTIM 121181-53-1
Price
US $1.10/g
Min. Order
1g
Purity
99.9%
Supply Ability
100 Tons min
Release date
2021-08-04

121181-53-1, FILGRASTIMRelated Search:


  • FILGRASTIM
  • n-l-methionyl-colony-stimulatingfactor(humanclone1034
  • Colony-stiMulating factor (huMan clone 1034), N-L-Methionyl- (9CI)
  • Filgrastim CRS
  • FILGRASTIM USP/EP/BP
  • Filgrastim DISCONTINUED
  • Figrastim
  • filgrastimconcentratedSolution
  • Filgrastim for Bioassay (96,815 IU) (COLD SHIPMENT REQUIRED)
  • Filgrastim System Suitability (COLD SHIPMENT REQUIRED) (1 mg)
  • 121181-53-1