ChemicalBook > CAS DataBase List > Zoxazolamine

Zoxazolamine

Product Name
Zoxazolamine
CAS No.
61-80-3
Chemical Name
Zoxazolamine
Synonyms
Zoxine;Flexin;Zoxamin;McN-485;Deflexol;Flexilon;usafma-12;NSC 24995;Contrazole;USAF ma-12
CBNumber
CB7464410
Molecular Formula
C7H5ClN2O
Formula Weight
168.58
MOL File
61-80-3.mol
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Zoxazolamine Property

Melting point:
181-184 °C(lit.)
Boiling point:
316.8±34.0 °C(Predicted)
Density 
1.4369 (rough estimate)
refractive index 
1.5618 (estimate)
storage temp. 
Keep in dark place,Sealed in dry,2-8°C
solubility 
DMSO, Methanol
pka
0.73±0.10(Predicted)
form 
Powder
color 
Light brown to yellow-brown
Merck 
13,10249
CAS DataBase Reference
61-80-3(CAS DataBase Reference)
NIST Chemistry Reference
Zoxazolamine(61-80-3)
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Safety

Hazard Codes 
Xn
Risk Statements 
20/21/22-36/37/38
Safety Statements 
26-36
WGK Germany 
3
RTECS 
DM4550000
HS Code 
29349990
Toxicity
LD50 in mice, rats (mg/kg): 376, 102 i.p.; 678, 730 orally (Cain, Roszkowski)
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
A45807
Product name
2-Amino-5-chlorobenzoxazole
Purity
97%
Packaging
5g
Price
$188
Updated
2024/03/01
Sigma-Aldrich
Product number
A45807
Product name
2-Amino-5-chlorobenzoxazole
Purity
97%
Packaging
1g
Price
$58.7
Updated
2023/06/20
Cayman Chemical
Product number
17565
Product name
Zoxazolamine
Purity
≥98%
Packaging
1g
Price
$32
Updated
2024/03/01
Cayman Chemical
Product number
17565
Product name
Zoxazolamine
Purity
≥98%
Packaging
5g
Price
$109
Updated
2024/03/01
Sigma-Aldrich
Product number
A45807
Product name
2-Amino-5-chlorobenzoxazole
Purity
97%
Packaging
25g
Price
$572
Updated
2024/03/01
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Zoxazolamine Chemical Properties,Usage,Production

Chemical Properties

LIGHT BROWN TO YELLOW-BROWN POWDER

Originator

Flexin ,McNeil,US,1956

Uses

sweetener

Uses

Zoxazolamine is a centrally acting myorelaxant; formerly used as an antispasmodic and uricosuric. Used as a tool for assessing hepatic cytochrome P-450 activity in rodents.

Definition

ChEBI: Zoxazolamine is a benzoxazole.

Manufacturing Process

To a solution of 106 g (0.74 mol) of 2-amino-4-chlorophenol in 500 ml of water containing 69 ml of concentrated hydrochloric acid (29.2 g, 0.8 mol) are added 60.8 g (0.8 mol) of ammonium thiocyanate. The solution is placed in an evaporating dish and heated on a steam bath for 5 hours. The solid which results is then removed from the concentrated solution by filtration, washed with a small amount of water and dried. The filtrate is placed in an evaporating dish and heated on a water bath for 2 hours. At the end of this time, the mixture is cooled, and the solid which precipitates out is removed by filtration. Both solid products are 5-chloro-2-hydroxyphenylthiourea melting at 157°C, and may be combined. The calculated N content for C 7 H 7 ClN 2 OS is 13.8; that found is 13.6.
To a solution of 10 g (0.05 mol) of 2-hydroxy-5-chlorophenylthiourea in 50 ml of methanol is added a solution of 11 g (0.04 mol) of ferric chloride hexahydrate in 50 ml of methanol. The initial purple-red color changes in a few minutes to amber. After stirring for one half hour, the solution is treated with 16.5 ml of 57% ammonium hydroxide solution (0.24 mol). A brown, flocculent precipitate of ferric sulfide appears. The mixture is then refluxed with stirring for one hour, cooled and centrifuged. The centrifugate is evaporated to dryness, and the residue is shaken with ether and water to separate the organic material from the ammonium chloride. The ether layer is extracted three times with 25 ml portions of 1 N hydrochloric acid. The acid solution is then poured into excess ammonium hydroxide, and the resulting solid collected, washed with water and dried. This gives a light tan solid melting at 183°C to 185°. The material is then dissolved in 25 ml of acetone and 50 ml of benzene are added. After treatment of the solution with activated charcoal, the light yellow solution is evaporated to 25 ml and cooled. The white crystals of 2-amino-5-chlorobenzoxazole which separate melt at 185°C to 186°C.

Therapeutic Function

Muscle relaxant, Uricosuric

Zoxazolamine Preparation Products And Raw materials

Raw materials

Preparation Products

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Zoxazolamine Suppliers

J & K SCIENTIFIC LTD.
Tel
010-82848833 400-666-7788
Fax
86-10-82849933
Email
jkinfo@jkchemical.com
Country
China
ProdList
94657
Advantage
76
Energy Chemical
Tel
021-021-58432009 400-005-6266
Fax
021-58436166
Email
sales8178@energy-chemical.com
Country
China
ProdList
44689
Advantage
61
Wuhan Chemwish Technology Co., Ltd
Tel
86-027-67849912
Fax
86-027-87531808
Email
sales@chemwish.com
Country
China
ProdList
35896
Advantage
56
Capot Chemical Co., Ltd
Tel
+86 (0) 571 85 58 67 18
Fax
0086-571-85864795
Email
sales@capotchem.com
Country
China
ProdList
18207
Advantage
66
Beijing Ouhe Technology Co., Ltd
Tel
010-82967028 13552068683
Fax
+86-10-82967029
Email
2355560935@qq.com
Country
China
ProdList
12390
Advantage
60
JinYan Chemicals(ShangHai) Co.,Ltd.
Tel
13817811078
Fax
86-021-50426522,50426273
Email
sales@jingyan-chemical.com
Country
China
ProdList
9976
Advantage
60
Shanghai Sinch Parmaceuticals Tech. Co. Ltd.
Tel
+86-21-54098501
Fax
+86-21-54096319
Email
sales@sinch.com.cn
Country
China
ProdList
11598
Advantage
64
Tetranov Biopharm
Tel
13526569071
Email
sales@leadmedpharm.com
Country
China
ProdList
7905
Advantage
64
Adamas Reagent, Ltd.
Tel
400-6009262 16621234537
Fax
021-64823266
Email
chenyj@titansci.com
Country
China
ProdList
14103
Advantage
59
Shanghai Longsheng chemical Co.,Ltd.
Tel
021-58099652-8005 13585536065
Fax
021-58099609
Email
bin.wu@shlschem.com
Country
China
ProdList
9809
Advantage
59
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View Lastest Price from Zoxazolamine manufacturers

Zhejiang J&C Biological Technology Co.,Limited
Product
Zoxazolamine 61-80-3
Price
US $0.00/gram
Min. Order
1gram
Purity
99%
Supply Ability
10kg
Release date
2022-02-17
Career Henan Chemical Co
Product
Zoxazolamine 61-80-3
Price
US $8.00/kg
Min. Order
1kg
Purity
99%
Supply Ability
10TON
Release date
2018-12-18

61-80-3, ZoxazolamineRelated Search:


  • 2-AMINO-5-CHLOROBENZOXAZOLE
  • usafma-12
  • Zoxamin
  • Zoxine
  • TIMTEC-BB SBB003874
  • ZOXAZOLAMINE
  • 2-Amino-5-chlorobenzoxazole,97%
  • 2-Amino-5-chlorobenzoxazoleZoxazolamine
  • 5-chlorobenzo[d]oxazol-2-aMine
  • 2-amino-5-chloro-benzoxazol
  • 2-Benzoxazolamine, 5-chloro-
  • 5-Chloro-1,3-benzoxazol-2-amine
  • 5-Chloro-2-benzoxazolamine
  • Benzoxazole, 2-amino-5-chloro-
  • Contrazole
  • Deflexol
  • Flexilon
  • Flexin
  • McN-485
  • USAF ma-12
  • 2-Benzoxazolamine, 5-chloro- (9CI)
  • NSC 24995
  • (5-chloro-1,3-benzoxazol-2-yl)amine
  • Zossazolamina [DCIT]
  • NSC 24995|||Contrazole
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