ERK Inhibitor
- Product Name
- ERK Inhibitor
- CAS No.
- 1049738-54-6
- Chemical Name
- ERK Inhibitor
- Synonyms
- ERK-IN-4;ERK Inhibitor - CAS 1049738-54-6 - Calbiochem;3-(2-aminoethyl)-5-[(4-ethoxyphenyl)methylene]-2,4-thiazolidinedione,monohydrochloride;(5Z)-3-(2-aminoethyl)-5-[(4-ethoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione:hydrochloride
- CBNumber
- CB13136749
- Molecular Formula
- C14H17ClN2O3S
- Formula Weight
- 328.81
- MOL File
- 1049738-54-6.mol
ERK Inhibitor Property
- storage temp.
- +2C to +8C
- solubility
- DMSO: 2 mg/ml
- form
- Light yellow solid
- color
- Off-white to yellow
N-Bromosuccinimide Price
- Product number
- 15944
- Product name
- ERK Inhibitor
- Purity
- ≥95%
- Packaging
- 500μg
- Price
- $32
- Updated
- 2024/03/01
- Product number
- 15944
- Product name
- ERK Inhibitor
- Purity
- ≥95%
- Packaging
- 1mg
- Price
- $50
- Updated
- 2024/03/01
- Product number
- 15944
- Product name
- ERK Inhibitor
- Purity
- ≥95%
- Packaging
- 5mg
- Price
- $117
- Updated
- 2024/03/01
- Product number
- 9473CW
- Product name
- ErkInhibitor
- Packaging
- 5mg
- Price
- $228
- Updated
- 2021/12/16
ERK Inhibitor Chemical Properties,Usage,Production
Description
ERK inhibitor is a cell-
General Description
A cell-permeable and reversible thiazolidinedione compound that displays anti-proliferative properties (IC50 ≤ 25 μM in HeLa, A549, and SUM-159 tumor cells). Preferentially binds to ERK2 with a KD of ~5 μM and prevents its interaction with protein substrates. Shown to block ERK-mediated phosphorylation of ribosomal S6 kinase-1 (RSK-1) and ternary complex factor Elk-1 in HeLa cells, while exhibiting little effect on ERK1/2 phosphorylation by MEK1/2.
Biochem/physiol Actions
Primary TargetERK
ERK Inhibitor Preparation Products And Raw materials
Raw materials
Preparation Products
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