ERK Inhibitor
- Product Name
- ERK Inhibitor
- CAS No.
- 1049738-54-6
- Chemical Name
- ERK Inhibitor
- Synonyms
- ERK-IN-4;ERK Inhibitor - CAS 1049738-54-6 - Calbiochem;3-(2-aminoethyl)-5-[(4-ethoxyphenyl)methylene]-2,4-thiazolidinedione,monohydrochloride;(5Z)-3-(2-aminoethyl)-5-[(4-ethoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione:hydrochloride
- CBNumber
- CB13136749
- Molecular Formula
- C14H17ClN2O3S
- Formula Weight
- 328.81
- MOL File
- 1049738-54-6.mol
ERK Inhibitor Property
- storage temp.
- +2C to +8C
- solubility
- DMSO: 2 mg/ml
- form
- Light yellow solid
- color
- Off-white to yellow
N-Bromosuccinimide Price
- Product number
- 15944
- Product name
- ERK Inhibitor
- Purity
- ≥95%
- Packaging
- 500μg
- Price
- $32
- Updated
- 2024/03/01
- Product number
- 15944
- Product name
- ERK Inhibitor
- Purity
- ≥95%
- Packaging
- 1mg
- Price
- $50
- Updated
- 2024/03/01
- Product number
- 15944
- Product name
- ERK Inhibitor
- Purity
- ≥95%
- Packaging
- 5mg
- Price
- $117
- Updated
- 2024/03/01
- Product number
- 9473CW
- Product name
- ErkInhibitor
- Packaging
- 5mg
- Price
- $228
- Updated
- 2021/12/16
ERK Inhibitor Chemical Properties,Usage,Production
Description
ERK inhibitor is a cell-
General Description
A cell-permeable and reversible thiazolidinedione compound that displays anti-proliferative properties (IC50 ≤ 25 μM in HeLa, A549, and SUM-159 tumor cells). Preferentially binds to ERK2 with a KD of ~5 μM and prevents its interaction with protein substrates. Shown to block ERK-mediated phosphorylation of ribosomal S6 kinase-1 (RSK-1) and ternary complex factor Elk-1 in HeLa cells, while exhibiting little effect on ERK1/2 phosphorylation by MEK1/2.
Biochem/physiol Actions
Primary TargetERK
ERK Inhibitor Preparation Products And Raw materials
Raw materials
Preparation Products
ERK Inhibitor Suppliers
- Tel
- 021-57171705 13817537615
- Fax
- QQ3095748324
- sales@run-biotech.com
- Country
- China
- ProdList
- 2427
- Advantage
- 58
- Tel
- 021-61415566 800-8193336
- orderCN@merckgroup.com
- Country
- China
- ProdList
- 51456
- Advantage
- 80
- Tel
- 16314854226
- info@bocsci.com
- Country
- United States
- ProdList
- 9923
- Advantage
- 65
- Tel
- 021-65675885 18964387627
- Fax
- 021-65675885
- info@efebio.com
- Country
- China
- ProdList
- 9806
- Advantage
- 58
- Tel
- 400-9205774
- sales@glpbio.cn
- Country
- China
- ProdList
- 6777
- Advantage
- 58
- Tel
- +1-781-999-5354 +1-00000000000
- marketing@targetmol.com
- Country
- United States
- ProdList
- 32165
- Advantage
- 58
- Tel
- 18818260767
- Fax
- QQ 3610331285
- sales@chemegen.com
- Country
- China
- ProdList
- 11217
- Advantage
- 58
- Tel
- 021-38015121 15000105423
- wulan@absin.cn
- Country
- China
- ProdList
- 24731
- Advantage
- 58
- Tel
- 021-69568360 18916172912
- order@med-bio.cn
- Country
- China
- ProdList
- 8140
- Advantage
- 58
- Tel
- +86-02787215551 +86-19945035818
- Fax
- 027-87215551
- 2936752263@qq.com
- Country
- China
- ProdList
- 7973
- Advantage
- 58