Synthesis methods Uses
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1-Bromo-4-iodobenzene

Synthesis methods Uses
Product Name
1-Bromo-4-iodobenzene
CAS No.
589-87-7
Chemical Name
1-Bromo-4-iodobenzene
Synonyms
P-BROMOIODOBENZENE;4-BROMOIODOBENZENE;4-BroMoiodoben;p-Bromiodobenzene;4-IODOBROMOBENZENE;p-Iodobromobenzene;4- Bromiodobenzene;1-Brom-4-iodbenzol;1-BROMO-IODOBENZENE;4-Bromophenyl iodide
CBNumber
CB4266086
Molecular Formula
C6H4BrI
Formula Weight
282.9
MOL File
589-87-7.mol
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1-Bromo-4-iodobenzene Property

Melting point:
89-91 °C(lit.)
Boiling point:
120-122 °C14 mm Hg(lit.)
Density 
2.2236 (rough estimate)
refractive index 
1.6618 (estimate)
Flash point:
120-122°C/14mm
storage temp. 
Store below +30°C.
solubility 
0.008g/l
form 
Crystalline Powder, Crystals or Needles
color 
White to brown
Water Solubility 
Insoluble in water.
Sensitive 
Light Sensitive
BRN 
1904545
InChI
1S/C6H4BrI/c7-5-1-3-6(8)4-2-5/h1-4H
InChIKey
UCCUXODGPMAHRL-UHFFFAOYSA-N
SMILES
Brc1ccc(I)cc1
CAS DataBase Reference
589-87-7(CAS DataBase Reference)
NIST Chemistry Reference
Benzene, 1-bromo-4-iodo-(589-87-7)
EPA Substance Registry System
Benzene, 1-bromo-4-iodo- (589-87-7)
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Safety

Hazard Codes 
Xi
Risk Statements 
36/37/38
Safety Statements 
26-36-37/39
WGK Germany 
3
Hazard Note 
Harmful/Light Sensitive
TSCA 
TSCA listed
HazardClass 
IRRITANT, LIGHT SENSITIVE, IRRITANT-HARMFUL
HS Code 
29036990
Storage Class
11 - Combustible Solids
Hazard Classifications
Eye Irrit. 2
Skin Irrit. 2
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H315Causes skin irritation

H319Causes serious eye irritation

Precautionary statements

P302+P352IF ON SKIN: wash with plenty of soap and water.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
238090
Product name
1-Bromo-4-iodobenzene
Purity
98%
Packaging
5g
Price
$31
Updated
2025/07/31
Sigma-Aldrich
Product number
238090
Product name
1-Bromo-4-iodobenzene
Purity
98%
Packaging
25g
Price
$147
Updated
2025/07/31
TCI Chemical
Product number
B0604
Product name
1-Bromo-4-iodobenzene
Packaging
25G
Price
$71
Updated
2025/07/31
TCI Chemical
Product number
B0604
Product name
1-Bromo-4-iodobenzene
Packaging
250G
Price
$425
Updated
2025/07/31
TRC
Product number
B683675
Product name
1-Bromo-4-iodobenzene
Packaging
5g
Price
$55
Updated
2021/12/16
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1-Bromo-4-iodobenzene Chemical Properties,Usage,Production

Synthesis methods

Industrial parabromoaniline is as raw material, by diazotization, iodo-synthesis of bromo iodobenzene. Preferred synthesis conditions: firstly 0.02mol parabromoaniline is dissolved in a mass fraction of 20% sulfuric acid medium, then reacts with 0.021molNaNO2 to generate bromophenyl diazonium sulfate at-10℃, and then chloroform and 0.021molKI is added into solution to process iodination reaction, after simple treatment bromo-iodobenzene crude product (which the bromo-iodobenzene HPLC purity 98.4%) is obtained, total yield after purification is 80%, increases by 15% than before improved. The product processes structural characterization by IR and 1HNMR. The improved method can greatly improve the purity of the crude product, this avoids the trouble of going through the column, this method is safe and easy to operate, easy to control the process, cost is lower, it is more suitable for the preparation of 1-Bromo-4-iodobenzene.
Unit: Heilongjiang University of Chemistry and Materials Science
Author: Guo Jing Bai Xuefeng Lvhong Fei

Uses

1. 1-Bromo-4-iodobenzene is used for organic synthesis.
2. Used as substrate for copper-free Sonogashira coupling reaction in aqueous acetone.
3. For the synthesis of β,β-dibromostyrene.

Chemical Properties

white to brown cryst. powder, crystals or needles

Uses

suzuki reaction

Uses

1-Bromo-4-iodobenzene has been employed:

  • as reagent for in situ desilylation and coupling of silylated alkynes
  • as starting reagent in the total syntheses of ent-conduramine A and ent-7-deoxypancratistatin (alkaloids)
  • as substrate in copper-free Sonogashira coupling in aqueous acetone
  • in synthesis of β,β,dibromostyrenes

General Description

Vapour pressure as a function of temperature for 1-bromo-4-iodobenzene has been studied using a diaphragm manometer and torsion mass-loss effusion.

Synthesis

The p-bromoiodobenzene was synthesized by diazotization and iodination using industrial p-bromoaniline as raw material. The better synthesis conditions: firstly, 0.02 mol of p-bromoaniline was dissolved in 20% sulfuric acid, and reacted with 0.021 mol of NaNO2 to form p-bromobenzene diazonium sulfate at -10 ??, and then chloroform and 0.021 mol of KI were added to the solution for iodine substitution, and then p-bromoiodobenzene was obtained as a crude product after simple post-processing (in which the purity was 98.4%), and the total yield after purification was 80%, which was better than that of the improved synthesis. 98.4%), and the total yield reached 80% after purification, which was 15% higher than that before improvement. The product was structurally characterized by IR and 1HNMR. The improved method greatly improved the purity of the crude product, avoided the trouble of passing through the column, was easy and safe to operate, easy to control the process, low cost, and more suitable for the preparation of p-bromoiodobenzene.
Unit??School of Chemistry, Chemical Engineering and Materials, Heilongjiang University
Author??Guo Jing, Bai Xuefeng, Lv Hongfei

1-Bromo-4-iodobenzene Preparation Products And Raw materials

Raw materials

Preparation Products

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1-Bromo-4-iodobenzene Suppliers

Jiangsu Aikon Biopharmaceutical R&D co.,Ltd.
Tel
025-66113011 17798518460
Fax
(1)02557626880
Email
cfzhang@aikonchem.com
Country
China
ProdList
19906
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55
Weifang QianJin Fine Chemical Co., Ltd.
Tel
18753684562
Fax
0536-8897109
Email
1577399715@qq.COM
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China
ProdList
1739
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Weifang Siyuan Chemical Co., Ltd.
Tel
0536-8888106 17663601818
Fax
0536-8888106
Email
2354379876@qq.com
Country
China
ProdList
245
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Suzhou chems bio-tech.co.,Ltd.
Tel
0512-67903504 13814824891
Fax
QQ604360797
Email
604360797@qq.com
Country
China
ProdList
399
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ChangShu HengYao Advanced Material Co.,Ltd.
Tel
0510-15312278075 15312278075
Email
xxl_hotmail@163.com
Country
China
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224
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NANJING SHUNXIANG PHARMACEUTICAL TECHNOLOGY CO.,LTD.
Tel
86819868 13951004015
Fax
025-86819859
Email
sales@jinchemical.com
Country
China
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25
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58
Zhengzhou Jicheng Chemical Technology Co., Ltd
Tel
15737124187; 15737124187
Email
1811685958@qq.com
Country
China
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304
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Shaanxi Lihe Tongchuang Chemical Technology Co., Ltd
Tel
029-81116050 17782851193
Email
168361757@qq.com
Country
China
ProdList
974
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J & K SCIENTIFIC LTD.
Tel
18210857532; 18210857532
Fax
86-10-82849933
Email
jkinfo@jkchemical.com
Country
China
ProdList
96815
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76
Sichuan Ruibo Technology Co., Ltd
Tel
+86-817-5586080
Fax
+86-817-5527378
Country
China
ProdList
42
Advantage
69
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View Lastest Price from 1-Bromo-4-iodobenzene manufacturers

Nanjing Shunxiang Pharmaceutical Technology Co.,Ltd.
Product
1-Bromo-4-iodobenzene 589-87-7
Price
US $0.00/kg
Min. Order
1kg
Purity
99%
Supply Ability
1
Release date
2025-09-26
Hebei Chuanghai Biotechnology Co., Ltd
Product
1-Bromo-4-iodobenzene 589-87-7
Price
US $1.00/KG
Min. Order
1KG
Purity
99%
Supply Ability
10 mt
Release date
2025-03-10
Speranza Chemical Co., Ltd.
Product
1-Bromo-4-iodobenzene 589-87-7
Price
US $25.00/KG
Min. Order
1KG
Purity
98%+
Supply Ability
300MT/year
Release date
2019-12-24

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