PROTAC ERRα Degrader-1 CAS#: 2306388-84-9

PROTAC ERRα Degrader-1 Basic information

Product Name:

PROTAC ERRα Degrader-1

Synonyms:

PROTAC ERRα Degrader-1
1-Piperazineacetamide, 4-[[(4R,5S)-4,5-bis(4-chlorophenyl)-4,5-dihydro-2-[4-methoxy-2-(1-methylethoxy)phenyl]-1H-imidazol-1-yl]carbonyl]-N-[2-[[(2E)-3-[4-[[2,4-bis(trifluoromethyl)phenyl]methoxy]-3-methoxyphenyl]-2-cyano-1-oxo-2-propen-1-yl]amino]ethyl]-2-oxo-

CAS:

2306388-84-9

MF:

C54H49Cl2F6N7O8

MW:

1108.91

Mol File:

2306388-84-9.mol

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PROTAC ERRα Degrader-1 Chemical Properties

Density: 1.38±0.1 g/cm3(Predicted)
storage temp.: Store at -20°C
solubility: Soluble in DMSO
pka: 11.80±0.46(Predicted)
form: Solid
color: White to off-white

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PROTAC ERRα Degrader-1 Usage And Synthesis

Description

ERRα Degrader-1 is a Novel PROTAC Estrogen-related Receptor α (ERRα) Degrader.

Description

ERRα Degrader-1 is a Novel PROTAC Estrogen-related Receptor α (ERRα) Degrader.

Uses

PROTAC ERRα Degrader-1 comprises a MDM2 ligand binding group, a linker and an estrogen-related receptor alpha (ERRa) binding group. PROTAC ERRα Degrader-1 is an PROTAC estrogen-related receptor alpha (ERRa) degrader[1].

IC 50

ERRα; MDM2

References

[1] Peng L, et al. Identification of New Small-Molecule Inducers of Estrogen-related Receptor α (ERRα) Degradation. ACS Med Chem Lett. 2019 Apr 12;10(5):767-772. DOI:10.1021/acsmedchemlett.9b00025

PROTAC ERRα Degrader-1Supplier

Sichuan Wei Keqi Biological Technology Co., Ltd.

Tel: 028-81700200 18116577057
Email: 3003855609@qq.com

Jilin Province Woda Biotechnology Co., Ltd.

Tel: 13504435624
Email: 1927928688@qq.com

TargetMol Chemicals Inc.

Tel: +1-781-999-5354; +17819995354
Email: marketing@targetmol.com

Beijing Jin Ming Biotechnology Co., Ltd.

Tel: 010-60605840 15801484223;
Email: psaitong@jm-bio.com

ShenZhen Trendseen Biological Technology Co.,Ltd.

Tel: 13417589054;
Email: trendseenbio@gmail.com

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